Product Name :
LY2119620
Description:
LY2119620 is a high-affinity muscarinic M2/M4 receptor agonist.
CAS:
886047-22-9
Molecular Weight:
437.94
Formula:
C19H24ClN5O3S
Chemical Name:
3-amino-5-chloro-N-cyclopropyl-4-methyl-6-[2-(4-methylpiperazin-1-yl)-2-oxoethoxy]thieno[2,3-b]pyridine-2-carboxamide
Smiles :
CN1CCN(CC1)C(=O)COC1=NC2SC(=C(N)C=2C(C)=C1Cl)C(=O)NC1CC1
InChiKey:
TYTGOXSAAQWLPJ-UHFFFAOYSA-N
InChi :
InChI=1S/C19H24ClN5O3S/c1-10-13-15(21)16(17(27)22-11-3-4-11)29-19(13)23-18(14(10)20)28-9-12(26)25-7-5-24(2)6-8-25/h11H,3-9,21H2,1-2H3,(H,22,27)
Purity:
≥98% (or refer to the Certificate of Analysis)
Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition :
Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.Tazemetostat medchemexpress
Shelf Life:
≥12 months if stored properly.Vadadustat custom synthesis
Stock Solution Storage:
0 – 4 oC for 1 month or refer to the Certificate of Analysis.
Additional information:
LY2119620 is a high-affinity muscarinic M2/M4 receptor agonist.|Product information|CAS Number: 886047-22-9|Molecular Weight: 437.94|Formula: C19H24ClN5O3S|Chemical Name: 3-amino-5-chloro-N-cyclopropyl-4-methyl-6-[2-(4-methylpiperazin-1-yl)-2-oxoethoxy]thieno[2,3-b]pyridine-2-carboxamide|Smiles: CN1CCN(CC1)C(=O)COC1=NC2SC(=C(N)C=2C(C)=C1Cl)C(=O)NC1CC1|InChiKey: TYTGOXSAAQWLPJ-UHFFFAOYSA-N|InChi: InChI=1S/C19H24ClN5O3S/c1-10-13-15(21)16(17(27)22-11-3-4-11)29-19(13)23-18(14(10)20)28-9-12(26)25-7-5-24(2)6-8-25/h11H,3-9,21H2,1-2H3,(H,22,27)|Technical Data|Appearance: Solid Power|Purity: ≥98% (or refer to the Certificate of Analysis)|Solubility: DMSO : 67.PMID:32811349 5 mg/mL (154.13 mM; Need ultrasonic).|Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis|Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.|Shelf Life: ≥12 months if stored properly.|Stock Solution Storage: 0 – 4 oC for 1 month or refer to the Certificate of Analysis.|Drug Formulation: To be determined|HS Tariff Code: 382200|How to use|In Vitro:|LY2119620 shows a modest allosteric agonism of 23.2±2.18% and 16.8±5.01% at the M2 and M4 receptors, respectively. Minimal allosteric agonism (Products are for research use only. Not for human use.|